Template:Relative affinities of noretynodrel, tibolone, and metabolites
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| Compound | Code name | PR | AR | ER | GR | MR | SHBG | CBG |
|---|---|---|---|---|---|---|---|---|
| Noretynodrel | – | 6 | 0 | 2 | 0 | 0 | 0 | 0 |
| Norethisterone (δ4-NYD) | – | 67–75 | 15 | 0 | 0–1 | 0–3 | 16 | 0 |
| 3α-Hydroxynoretynodrel | – | ? | ? | ? | ? | ? | ? | ? |
| 3β-Hydroxynoretynodrel | – | ? | ? | ? | ? | ? | ? | ? |
| Ethinylestradiol | – | 15–25 | 1–3 | 112 | 1–3 | <1 | 0.18 | <0.1 |
| Tibolone (7α-Me-NYD) | ORG-OD-14 | 6 | 6 | 1 | ? | ? | ? | ? |
| Δ4-Tibolone | ORG-OM-38 | 90 | 35 | 1 | 0 | 2 | 1 | 0 |
| 3α-Hydroxytibolone | ORG-4094 | 0 | 3 | 4–6 | 0 | ? | ? | ? |
| 3β-Hydroxytibolone | ORG-301260 | 0 | 4 | 3–29 | 0 | ? | ? | ? |
| 7α-Methylethinylestradiol | – | ? | ? | ? | ? | ? | ? | ? |
| Notes: Values are percentages (%). Reference ligands (100%) were promegestone for the PR, metribolone for the AR, E2 for the ER, DEXA for the GR, aldosterone for the MR, DHT for SHBG, and cortisol for CBG. Sources: [1][2][3][4][5][6] | ||||||||
Template documentationReferences
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